Caffeine - instruction , application reviews


1. Pharmacological Effects of Caffeine

2. Product form

3. Indications Caffeine

4. Dosing Caffeine

5. Side effects Caffeine

6. Overdose

7. Contraindications Caffeine

8. Drug interactions Caffeine

9. Cautions

10. shelf life

Caffeine - a drug that stimulates mental activity.

Pharmacological Effects of Caffeine Caffeine

drug sodium benzoate - a tool that helps to reduce sleepiness and fatigue, stimulating effect on human mental activity, as well as his mental and physical performance.

Caffeine is known for its aphrodisiac properties, aimed at performance respiratory and vasomotor centers, at enhancing cardiac function, as well as dilation of the blood vessels of the muscles, brain, heart, kidneys and narrowing of blood vessels of the abdominal cavity.

Applied elderly patients benzoate Caffeine has a significant effect on their sleep: it slows the onset and reduces the overall duration of sleep and increased frequency of awakenings.

Premature babies this drug reduces the partial pressure of carbon dioxide, eliminating the periodic breathing and increases the amount of ventilation, without affecting heart rate.

Product form Available Caffeine tablets and capsules (solutions for subcutaneous and subconjunctival injection).

Indications Caffeine Caffeine

Apply benzoate in reducing mental and physical performance, with drowsiness, headache vascular character, moderate hypotension, respiratory depression and enuresis.The tool is also effective to restore the required level of pulmonary ventilation after suffering anesthesia.

In ophthalmology Caffeine is used in retinal detachment and lowering the tone after surgery on the eye.

addition, the drug is used in the case of depression of the central nervous system caused by drug poisoning and fatty substances, primarily with alcohol intoxication.

In cosmetology widely used mixture of caffeine and Kapsikama as an effective remedy for anti-cellulite body wraps.

Dosing Caffeine

Adults take caffeine tablets to 50-100 mg 2-3 times per day.Children drug is administered in a dosage of 30-75 mg twice or thrice a day.Caffeine is not recommended to be taken before bedtime.Caffeine

in ampoules, 1 ml administered subcutaneously.The maximum single dose - 0.4 grams daily and - less than 1 gram.Children are 10% caffeine solution in ampoules of 0.25-1 ml.

administration used in ophthalmology 10% solution of caffeine by injection under the conjunctiva at a dose of 0.3 ml once a day.Multiplicity of dosing depends on the intraocular pressure and the ocular anterior chamber depth.

Anti-cellulite wrapping "Caffeine Kapsikam" is performed as follows: A mixture of 4 vials of caffeine Kapsikam ointment (approximately 2 cm) and baby oil (about 4 cm).The mixture of caffeine and Kapsikama applied to the "problem" areas of the body, cover with cling film and kept on the skin for 3 hours.An hour before applying application, during the procedure, and within 2 hours after it is advisable not to drink or eat.Duration of the course - 10 procedures.

Side effects Caffeine

Since the cardiovascular system: heart palpitations, increased blood pressure, arrhythmia, tachycardia.

From the nervous system: anxiety, anxiety, agitation, headache, tremors, dizziness, tachypnea, seizures, insomnia, increased reflexes.

From the digestive system: exacerbation of peptic ulcer, vomiting, nausea.

Long-term use caffeine benzoate can cause addiction and dependence on the drug.

Anti-cellulite wrap with caffeine and Kapsikama accompanied by a burning sensation on the skin during the whole procedure.


Caffeine in doses of 300 mg per day or more can cause the following symptoms: anxiety, agitation, delirium, confusion, restlessness, gastralgia, agitation, tachycardia, dehydration, hyperthermia, arrhythmias, headache, frequent urination, increasedpain or tactile sensitivity, muscle twitching or tremors, nausea and vomiting, seizures, ringing in the ears.

Treatment: gastric lavage, if adopted in recent Caffeine 4 hours a dosage greater than 15 mg / kg body weight and this was not vomiting;laxatives drugs and activated carbon;in the presence of hemorrhagic gastritis carried administering antacids and gastric lavage ice 0.9% solution of NaCl;maintenance of oxygenation and ventilation;when administered intravenously seizures phenobarbital, phenytoin, or diazepam;maintaining salts and water balance.Newborn children performed exchange transfusion if necessary.

Contraindications Caffeine

forbidden to take caffeine tablets, as well as do caffeine injection in vials at the following illnesses: hypertension, anxiety disorders, organic disorders of the cardiovascular system, frequent ventricular premature beats, paroxysmal tachycardia, sleep disturbances and hypersensitivity to the drug.

Caffeine is not indicated for children under 12 years.

wary drug should be used for older people, during pregnancy and lactation, as well as in patients with glaucoma, epilepsy and a tendency to seizures.

Drug Interactions Caffeine

When combined with caffeine decreases the effectiveness of sleeping pills and drugs for anesthesia.

While the use of caffeine-containing medications may be a strengthening of action of naproxen, salicylamide-antipyretics and analgesics.

One-time intake of caffeine and acetylsalicylic acid can increase its bioavailability, the rate of absorption and concentration in blood plasma.

Mexiletine decreases caffeine clearance and increases its concentration in the blood.

methoxsalen slows the process of removing caffeine from the body with the development of its toxic effect and increased effect.

terbinafine, fluconazole and ketoconazole caused a slight increase in the content of caffeine in the blood.

With simultaneous use of ergotamine and caffeine speeds up the process of absorption of the latter.


Abrupt discontinuation of caffeine can cause central nervous system enhancement and inhibition cause drowsiness and depression.Effect of the drug on the CNS depends primarily on the type of the nervous system, and may appear as a brake and the excitation of higher nervous activity.Since the effects of caffeine on blood pressure is made up of the cardiac and vascular components, as a result may develop as the stimulation of cardiac activity, and weakly expressed her depression.

When apnea in newborn babies in the postoperative period is used Caffeine Caffeine citrate or just, but not caffeine sodium benzoate.

excessive use of caffeine during pregnancy may provoke spontaneous abortions, fetal arrhythmia in, slowing its prenatal development, disturbance and retardation of skeletal development.

Shelf life Shelf life

Caffeine Caffeine tablets and ampoules of 5 years.


Product description posted on this page is a supplement and a simplified version of the official version of the annotations to the drug.The information is provided for informational purposes only and is not a guide to self-medication.Before using the product you should consult with a specialist and to get acquainted with the instructions approved by the manufacturer.

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